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YM-254890

In stock
Catalog ID
253-00633
$1,683.00
Sku
253-00633
Details

for Cellbiology

This product is for research use only. Do not administer it to humans.

Trimeric G proteins, Gq family specific inhibitor.

This is a cyclic depsipeptide isolated from a soil bacterium Chromobacterium sp. QS3666 strain and has a cyclic peptide structure composed of unique amino acids differing from normal amino acids.

It specifically inhibits signals mediated by Gq family of trimeric G proteins, Gq, G11 and G14, which are involved in elevated Ca2+ level among about 20 types of G proteins, by acting on GDT/GTP exchange reaction. It is a first membrane permeable compound particularly inhibiting Gq signal and a useful tool for a study analyzing Gq signals.

  • Specifically inhibits signals mediated by Gαaq, Gα11, and Gα14

  • Acts in both in vivo and in vitro systems

How to use: dissolve it in DMSO at 1-10 mmol/L to prepare stock solution. In use, accordingly dilute it with an experimental solution.

  • Go through the stock solution as soon as possible.

Precautions for Use: Packed on argon gas
Appearance: White - pale brown, crystalline powder - powder
Specification Assay: 95.0+% (HPLC)
CAS RN: 568580-02-9
Molecular Formula: C46H69N7O15
Molecular Weight: 960.08

 

Made by FUJIFILM Wako Pure Chemical Corporation and distributed by FUJIFILM Irvine Scientific

  • For research use only. Not for use in diagnostic procedures.

  • Product content may differ from the actual image due to minor specification changes etc.

  • If the revision of product standards and packaging standards has been made, there is a case where the actual product specifications and images are different.

Specifications

Storage
Keep at 2-10°C
Product Specifications
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